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Waleed Zalloum
Waleed Zalloum
Assistant professor of medicinal chemistry and drug design
Verifierad e-postadress på aum.edu.jo
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Discovery of new potent human protein tyrosine phosphatase inhibitors via pharmacophore and QSAR analysis followed by in silico screening
MO Taha, Y Bustanji, AG Al-Bakri, AM Yousef, WA Zalloum, IM Al-Masri, ...
Journal of Molecular Graphics and Modelling 25 (6), 870-884, 2007
1052007
Design, synthesis and structure-activity relationships of 4-phenyl-1H-1, 2, 3-triazole phenylalanine derivatives as novel HIV-1 capsid inhibitors with promising antiviral …
L Sun, T Huang, A Dick, ME Meuser, WA Zalloum, CH Chen, X Ding, ...
European Journal of Medicinal Chemistry 190, 112085, 2020
802020
Discovery of potent inhibitors of pseudomonal quorum sensing via pharmacophore modeling and in silico screening
MO Taha, AG Al-Bakri, WA Zalloum
Bioorganic & medicinal chemistry letters 16 (22), 5902-5906, 2006
642006
Discovery of phenylalanine derivatives as potent HIV-1 capsid inhibitors from click chemistry-based compound library
G Wu, WA Zalloum, ME Meuser, L Jing, D Kang, CH Chen, Y Tian, ...
European journal of medicinal chemistry 158, 478-492, 2018
562018
Discovery of novel 1, 4-disubstituted 1, 2, 3-triazole phenylalanine derivatives as HIV-1 capsid inhibitors
X Jiang, G Wu, WA Zalloum, ME Meuser, A Dick, L Sun, CH Chen, D Kang, ...
RSC advances 9 (50), 28961-28986, 2019
482019
Design, synthesis, and mechanism study of benzenesulfonamide-containing phenylalanine derivatives as novel HIV-1 capsid inhibitors with improved antiviral activities
L Sun, A Dick, ME Meuser, T Huang, WA Zalloum, CH Chen, ...
Journal of medicinal chemistry 63 (9), 4790-4810, 2020
462020
Novel urate transporter 1 (URAT1) inhibitors: a review of recent patent literature (2016–2019)
Y Dong, T Zhao, W Ai, WA Zalloum, D Kang, T Wu, X Liu, P Zhan
Expert Opinion on Therapeutic Patents 29 (11), 871-879, 2019
432019
Novel in vitro and in vivo anti-Helicobacter pylori effects of pomegranate peel ethanol extract
A Mayyas, M Abu-Sini, R Amr, RT Akasheh, W Zalloum, A Khdair, ...
Veterinary World 14 (1), 120, 2021
202021
Design, synthesis, and mechanism study of dimerized phenylalanine derivatives as novel HIV-1 capsid inhibitors
X Zhang, L Sun, ME Meuser, WA Zalloum, S Xu, T Huang, S Cherukupalli, ...
European journal of medicinal chemistry 226, 113848, 2021
182021
Discovery of Novel Dihydrothiopyrano[4,3-d]pyrimidine Derivatives as Potent HIV-1 NNRTIs with Significantly Reduced hERG Inhibitory Activity and Improved …
Z Wang, WA Zalloum, W Wang, X Jiang, E De Clercq, C Pannecouque, ...
Journal of Medicinal Chemistry 64 (18), 13658-13675, 2021
152021
Homology modeling of MCH1 receptor and validation by docking/scoring and protein-aligned CoMFA
A Abu-Hammad, WA Zalloum, H Zalloum, G Abu-Sheikha, MO Taha
European journal of medicinal chemistry 44 (6), 2583-2596, 2009
152009
Design, synthesis, and mechanistic investigations of phenylalanine derivatives containing a benzothiazole moiety as HIV-1 capsid inhibitors with improved metabolic stability
S Xu, L Sun, A Dick, WA Zalloum, T Huang, ME Meuser, X Zhang, Y Tao, ...
European journal of medicinal chemistry 227, 113903, 2022
142022
The effect of ferrous ions, calcium ions and citric acid on absorption of ciprofloxacin across caco-2 cells: practical and structural approach
D El-Sabawi, R Abu-Dahab, WA Zalloum, F Ijbara, II Hamdan
Drug Development and Industrial Pharmacy 45 (2), 292-303, 2019
142019
The effect of Ginkgo biloba and psycho-education on stress, anxiety and fatigue among refugees
AM Alsmadi, LI Tawalbeh, OS Gammoh, MQ Shawagfeh, W Zalloum, ...
Proceedings of Singapore Healthcare 27 (1), 26-32, 2018
142018
Fluorescent probe for detection of bacteria: conformational trigger upon bacterial reduction of an azo bridge
NJW Rattray, WA Zalloum, D Mansell, J Latimer, CH Schwalbe, AJ Blake, ...
Chemical communications 48 (51), 6393-6395, 2012
142012
Chemical and bacterial reduction of azo-probes: monitoring a conformational change using fluorescence spectroscopy
NJW Rattray, WA Zalloum, D Mansell, J Latimer, M Jaffar, EV Bichenkova, ...
Tetrahedron 69 (13), 2758-2766, 2013
122013
Discovery of novel “Dual-site” binding oseltamivir derivatives as potent influenza virus neuraminidase inhibitors
W Ai, J Zhang, WA Zalloum, R Jia, S Cherukupalli, X Ding, Z Sun, L Sun, ...
European Journal of Medicinal Chemistry 191, 112147, 2020
112020
Comparative molecular dynamics simulation of aggregating and non‐aggregating inhibitor solutions: understanding the molecular basis of promiscuity
MA Ghattas, RA Bryce, S Al Rawashdah, N Atatreh, WA Zalloum
ChemMedChem 13 (6), 500-506, 2018
102018
Perception, knowledge and attitude towards influenza vaccine during COVID-19 pandemic in Jordanian population
WA Zalloum, ER Elayeh, BAH Ali, N Zalloum
European Journal of Integrative Medicine 49, 102100, 2022
92022
Discovery and optimizing polycyclic pyridone compounds as anti-HBV agents
F Wei, D Kang, S Cherukupalli, WA Zalloum, T Zhang, X Liu, P Zhan
Expert Opinion on Therapeutic Patents 30 (9), 715-721, 2020
72020
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Artiklar 1–20